Lipid nanoparticles for transdermal delivery of flurbiprofen: formulation, in vitro, ex vivo and in vivo studies
2009

Lipid Nanoparticles for Transdermal Delivery of Flurbiprofen

Sample size: 6 publication 10 minutes Evidence: moderate

Author Information

Author(s): Bhaskar Kesavan, Anbu Jayaraman, Ravichandiran Velayutham, Venkateswarlu Vobalaboina, Rao Yamsani Madhusudan

Primary Institution: Kakatiya University

Hypothesis

The study aims to develop lipid nanoparticles for effective transdermal delivery of flurbiprofen.

Conclusion

The study found that both SLN and NLC formulations provided sustained drug release and improved bioavailability of flurbiprofen compared to oral administration.

Supporting Evidence

  • The Cmax of the NLC formulation was significantly higher than that of the SLN formulation.
  • The bioavailability of flurbiprofen increased by 4.4 times with the gel formulations compared to oral administration.
  • Both SLN and NLC formulations showed sustained drug release over 24 hours.

Takeaway

Researchers created special tiny particles to help deliver a pain medicine through the skin, which worked better than taking it by mouth.

Methodology

The study involved preparing lipid nanoparticles, incorporating them into hydrogels, and testing their drug release and skin permeation in rats.

Limitations

The study was conducted on rats, and results may not directly translate to humans.

Participant Demographics

Adult male Wistar albino rats weighing 230-250 g were used for in vivo studies.

Statistical Information

P-Value

p<0.01

Statistical Significance

p<0.01

Digital Object Identifier (DOI)

10.1186/1476-511X-8-6

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