Regulation of Bestrophins by Ca2+: A Theoretical and Experimental Study
2009

How Calcium Affects Bestrophins

publication 10 minutes Evidence: moderate

Author Information

Author(s): Kranjc Agata, Grillo Federico W., Rievaj Juraj, Boccaccio Anna, Pietrucci Fabio, Menini Anna, Carloni Paolo, Anselmi Claudio

Primary Institution: International School for Advanced Studies (SISSA/ISAS), Trieste, Italy

Hypothesis

The Asp-rich domain of bestrophins is involved in Ca2+ binding and activation.

Conclusion

The study confirms that mutations in the Asp-rich domain of bestrophins significantly affect their function and Ca2+-activated Cl− currents.

Supporting Evidence

  • Molecular dynamics simulations identified key residues in the Asp-rich domain that bind Ca2+.
  • Electrophysiological experiments confirmed that mutations in the Asp-rich domain affect Ca2+-activated Cl− currents.
  • The study suggests that at least two Ca2+-binding sites are present in the Asp-rich domain.

Takeaway

Bestrophins are proteins that help control chloride ions in cells, and this study shows how calcium affects their function by binding to specific parts of the protein.

Methodology

The study used molecular dynamics simulations and electrophysiological experiments to analyze the effects of mutations in the Asp-rich domain of bestrophins.

Limitations

The lack of structural information about the transmembrane region of the channel limits the understanding of how Ca2+ binding affects channel gating.

Statistical Information

P-Value

p<0.002

Statistical Significance

p<0.05

Digital Object Identifier (DOI)

10.1371/journal.pone.0004672

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