Acquisition of platinum drug resistance and platinum cross resistance patterns in a panel of human ovarian carcinoma xenografts
1993

Platinum Drug Resistance in Ovarian Cancer Models

Sample size: 6 publication Evidence: moderate

Author Information

Author(s): M. Jones, J. Siracky, L.R. Kelland, K.R. Harrap

Primary Institution: The Institute of Cancer Research

Hypothesis

Can human ovarian carcinoma xenografts develop resistance to platinum-based drugs?

Conclusion

The study established that resistance to platinum drugs can be generated in human ovarian carcinoma xenografts, with observed cross-resistance patterns.

Supporting Evidence

  • Resistance was generated to cisplatin, carboplatin, iproplatin, and tetraplatin.
  • Four tumors showed complete cross-resistance to the remaining platinum agents.
  • One line retained sensitivity to cisplatin and carboplatin despite resistance to iproplatin.

Takeaway

Researchers found that some ovarian cancer tumors can become resistant to chemotherapy drugs, making them harder to treat. They created models to study this resistance.

Methodology

The study used six human ovarian carcinoma xenografts to establish resistance to various platinum drugs through in vivo and in vitro treatments.

Limitations

The study primarily focused on a limited number of tumor lines and may not represent all ovarian cancers.

Participant Demographics

Tumor lines derived from previously untreated and treated patients.

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