Inhibition of PI3K Prevents the Proliferation and Differentiation of Human Lung Fibroblasts into Myofibroblasts: The Role of Class I P110 Isoforms PI3K in Fibroblasts Transformation/Proliferation
2011

Inhibition of PI3K Prevents Lung Fibroblast Growth

Sample size: 5 publication Evidence: moderate

Author Information

Author(s): Conte Enrico, Fruciano Mary, Fagone Evelina, Gili Elisa, Caraci Filippo, Iemmolo Maria, Crimi Nunzio, Vancheri Carlo

Primary Institution: Department of Clinical and Molecular Biomedicine, University of Catania, Catania, Italy

Hypothesis

The study investigates the role of the PI3K/Akt pathway in the proliferation and differentiation of human lung fibroblasts induced by TGF-β.

Conclusion

Inhibiting the PI3K pathway can prevent the proliferation and differentiation of lung fibroblasts into myofibroblasts, suggesting potential therapeutic targets for idiopathic pulmonary fibrosis.

Supporting Evidence

  • The pan-inhibitor of PI3Ks LY294002 abrogated TGF-β-induced increases in cell proliferation.
  • PI3K p110δ and p110γ were found to be functionally expressed in human lung fibroblasts.
  • Selective inhibitors demonstrated a major role of p110γ and p110α in TGF-β-induced fibroblast proliferation.

Takeaway

This study shows that blocking a specific pathway in lung cells can stop them from growing too much, which is important for treating a serious lung disease.

Methodology

The study used ex-vivo cultures of human lung fibroblasts and various PI3K inhibitors to assess their effects on cell proliferation and differentiation.

Participant Demographics

Human lung fibroblasts were derived from surgical lung specimens of patients undergoing resective surgery.

Statistical Information

P-Value

p<0.05

Statistical Significance

p<0.05

Digital Object Identifier (DOI)

10.1371/journal.pone.0024663

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