Catalytic synthesis of (E)-α,β-unsaturated esters from aldehydes and 1,1-diethoxyethylene
2009

Synthesis of α,β-unsaturated esters from aldehydes

publication Evidence: moderate

Author Information

Author(s): Manzano Rubén, Ozores Lidia, Job Andreas, Rodefeld Lars, List Benjamin, Clayden Jonathan

Primary Institution: Max-Planck-Institut für Kohlenforschung

Hypothesis

Can we develop a new catalytic method to synthesize α,β-unsaturated esters from aldehydes with high yields and selectivity?

Conclusion

A new catalytic method using boronic acids allows for the efficient synthesis of α,β-unsaturated esters from aldehydes with high yields.

Supporting Evidence

  • The new method achieved a yield of 98% for the synthesis of α,β-unsaturated esters.
  • Boronic acids were found to be the most effective catalysts in the reaction.
  • The procedure is applicable to both aromatic and aliphatic aldehydes.

Takeaway

Scientists found a new way to make a special type of chemical called α,β-unsaturated esters using simple ingredients and a special helper called a catalyst.

Methodology

The study involved the use of boronic acid as a catalyst to condense aldehydes with ketene diethyl acetal under specific conditions.

Digital Object Identifier (DOI)

10.3762/bjoc.5.3

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