Phosphodiesterase 4 inhibition but not beta-adrenergic stimulation suppresses tumor necrosis factor-alpha release in peripheral blood mononuclear cells in septic shock
2008

PDE4 Inhibition Reduces Inflammation in Septic Shock

Sample size: 40 publication 10 minutes Evidence: moderate

Author Information

Author(s): Link Andreas, Selejan Simina, Maack Christoph, Lenz Monika, Böhm Michael

Primary Institution: Klinik für Innere Medizin III, Universität des Saarlandes

Hypothesis

Is beta-adrenergic receptor downregulation in septic shock blunting the anti-inflammatory effects of catecholamines?

Conclusion

In septic shock, PDE4 inhibitors can maintain anti-inflammatory effects despite the downregulation of beta-adrenergic receptors.

Supporting Evidence

  • In septic shock, the anti-inflammatory effects of catecholamines are blunted by downregulation of beta2-adrenergic receptors.
  • PDE4 inhibitors maintain their anti-inflammatory efficacy in CD14+ monocytes despite beta-adrenergic downregulation.
  • The study involved 20 healthy volunteers and 20 patients with septic shock.

Takeaway

In patients with septic shock, the usual way that certain medicines help reduce inflammation doesn't work as well, but a different type of medicine can still help.

Methodology

The study involved in vitro stimulation of peripheral blood mononuclear cells from healthy volunteers and septic shock patients, analyzing TNF-α production and receptor expression.

Limitations

The study lacks data on PDE4 levels in monocytes from control subjects and septic patients.

Participant Demographics

20 healthy volunteers (median age 49) and 20 patients with septic shock (median age 52, 10 females and 10 males).

Statistical Information

P-Value

p<0.001

Statistical Significance

p<0.001

Digital Object Identifier (DOI)

10.1186/cc7158

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