NMR studies of anion-induced conformational changes in diindolylureas and diindolylthioureas
2011

NMR Studies of Anion-Induced Changes in Diindolylureas and Diindolylthioureas

publication Evidence: moderate

Author Information

Author(s): Makuc Damjan, Hiscock Jennifer R, Light Mark E, Gale Philip A, Plavec Janez

Primary Institution: Slovenian NMR Centre, National Institute of Chemistry

Hypothesis

The conformational properties of diindolylureas and diindolylthioureas change upon binding with anions.

Conclusion

The study found that anion binding causes significant conformational changes in diindolylureas and diindolylthioureas, with the syn–syn conformer being preferred in anion-receptor complexes.

Supporting Evidence

  • The anti–anti conformer was predominant in the absence of anions.
  • Strong deshielding of ureido protons was observed upon the addition of acetate, benzoate, bicarbonate, and dihydrogen phosphate.
  • Binding of oxo-anions caused conformational changes along the C7–N7α bonds.

Takeaway

This study looks at how certain chemical compounds change shape when they interact with different anions, which are negatively charged particles.

Methodology

The conformational properties were studied using heteronuclear NMR spectroscopy and quantum mechanics calculations.

Limitations

The study faced challenges in analyzing conformational changes for some compounds due to broad and overlapped NMR signals.

Digital Object Identifier (DOI)

10.3762/bjoc.7.140

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