Pharmacological Blockade of TRPM8 Ion Channels Alters Cold and Cold Pain Responses in Mice
2011

How a Drug Affects Cold Sensation in Mice

Sample size: 4 publication 10 minutes Evidence: high

Author Information

Author(s): Wendy M. Knowlton, Richard L. Daniels, Radhika Palkar, Daniel D. McCoy, David D. McKemy

Primary Institution: University of Southern California

Hypothesis

The study investigates the effects of a TRPM8 antagonist on cold sensation and thermoregulation in mice.

Conclusion

The TRPM8 antagonist PBMC significantly alters cold sensation and thermoregulation in mice.

Supporting Evidence

  • PBMC selectively blocks TRPM8 activity in vitro and in vivo.
  • PBMC administration resulted in dose-dependent hypothermia in wildtype mice.
  • TRPM8-knockout mice showed no response to PBMC treatment.

Takeaway

Researchers tested a drug that changes how mice feel cold, and it worked really well, making them less sensitive to cold temperatures.

Methodology

The study used calcium microfluorimetry and whole-cell voltage clamp recordings to assess the effects of PBMC on TRPM8 channels in vitro and in vivo.

Limitations

The study did not test higher doses of PBMC due to significant effects on thermoregulation.

Participant Demographics

Adult mice aged at least eight weeks, including wildtype and TRPM8-knockout mice.

Statistical Information

P-Value

p<0.001

Statistical Significance

p<0.001

Digital Object Identifier (DOI)

10.1371/journal.pone.0025894

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