Effect of Sulindac Sulfide on Metallohydrolases in the Human Colon Cancer Cell Line HT-29
2011

Effects of Sulindac on Colon Cancer Cells

publication Evidence: moderate

Author Information

Author(s): Hector Guillen-Ahlers, Jiangning Tan, Francis J. Castellino, Victoria A. Ploplis

Primary Institution: University of Notre Dame

Hypothesis

Does sulindac treatment affect metallohydrolases in human colon cancer cells?

Conclusion

Sulindac sulfide effectively downregulated MMP7 expression and activity in HT-29 human colon cancer cells.

Supporting Evidence

  • Sulindac sulfide significantly increased cell death in HT-29 cells.
  • MMP7 expression was downregulated by sulindac sulfide treatment.
  • The study shows that sulindac's effects in mice may be relevant to human colon cancer.

Takeaway

Sulindac, a common anti-inflammatory drug, can help reduce a protein linked to colon cancer in human cells.

Methodology

HT-29 cells were treated with sulindac and its metabolites, and MMP7 expression was measured using RT-PCR and Western blotting.

Limitations

The study primarily focuses on a single cell line and may not fully represent in vivo conditions.

Statistical Information

P-Value

p=0.000001

Statistical Significance

p<0.05

Digital Object Identifier (DOI)

10.1371/journal.pone.0025725

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