Meta-metallation of N,N-dimethylaniline: Contrasting direct sodium-mediated zincation with indirect sodiation-dialkylzinc co-complexation
2011

Meta-Metallation of N,N-Dimethylaniline

publication 10 minutes Evidence: high

Author Information

Author(s): David R. Armstrong, Liam Balloch, Eva Hevia, Alan R. Kennedy, Robert E. Mulvey, Charles T. O'Hara, Stuart D. Robertson, Victor Snieckus

Primary Institution: University of Strathclyde

Hypothesis

Can sodium-mediated zincation lead to meta-metallation of N,N-dimethylaniline?

Conclusion

The study demonstrates that sodium-mediated zincation can selectively produce the meta-isomer of N,N-dimethylaniline.

Supporting Evidence

  • The reaction of N,N-dimethylaniline with sodium TMP-zincate produced a mixture of ortho-, meta-, and para-regioisomers.
  • The meta-isomer was isolated in reasonable yields in a clean, pure crystalline form.
  • DFT calculations supported the experimental findings, indicating that the meta-isomer is the energetically preferred product.

Takeaway

This research shows how a special chemical reaction can change where a metal attaches to a molecule, making it possible to create new types of compounds.

Methodology

The study involved synthesizing and characterizing various organometallic complexes through reactions of N,N-dimethylaniline with sodium TMP-zincate and other reagents, followed by NMR and X-ray crystallography analysis.

Limitations

The study may be limited by the stability of the intermediates and the conditions required for the reactions.

Digital Object Identifier (DOI)

10.3762/bjoc.7.144

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